Partner ID 1558
Name Transient receptor potential cation channel subfamily V member 1
Synonyms 3324
Gene name TRPV1
General function Involved in ion channel activity
Specific function Receptor-activated non-selective calcium permeant cation channel involved in detection of noxious chemical and thermal stimuli. Seems to mediate proton influx and may be involved in intracellular acidosis in nociceptive neurons. May be involved in mediation of inflammatory pain and hyperalgesia. Sensitized by a phosphatidylinositol second messenger system activated by receptor tyrosine kinases, which involves PKC isozymes and PCL
Gene sequence + ...

ATGAAGAAATGGAGCAGCACAGACTTGGGGGCAGCTGCGGACCCACTCCAAAAGGACACCTGCCCAGACCCCCTGGATGGAGACCCTAACTCCAGGCCACCTCCAGCCAAGCCCCAGCTCTCCACGGCCAAGAGCCGCACCCGGCTCTTTGGGAAGGGTGACTCGGAGGAGGCTTTCCCGGTGGATTGCCCTCACGAGGAAGGTGAGCTGGACTCCTGCCCGACCATCACAGTCAGCCCTGTTATCACCATCCAGAGGCCAGGAGACGGCCCCACCGGTGCCAGGCTGCTGTCCCAGGACTCTGTCGCCGCCAGCACCGAGAAGACCCTCAGGCTCTATGATCGCAGGAGTATCTTTGAAGCCGTTGCTCAGAATAACTGCCAGGATCTGGAGAGCCTGCTGCTCTTCCTGCAGAAGAGCAAGAAGCACCTCACAGACAACGAGTTCAAAGACCCTGAGACAGGGAAGACCTGTCTGCTGAAAGCCATGCTCAACCTGCACGACGGACAGAACACCACCATCCCCCTGCTCCTGGAGATCGCGCGGCAAACGGACAGCCTGAAGGAGCTTGTCAACGCCAGCTACACGGACAGCTACTACAAGGGCCAGACAGCACTGCACATCGCCATCGAGAGACGCAACATGGCCCTGGTGACCCTCCTGGTGGAGAACGGAGCAGACGTCCAGGCTGCGGCCCATGGGGACTTCTTTAAGAAAACCAAAGGGCGGCCTGGATTCTACTTCGGTGAACTGCCCCTGTCCCTGGCCGCGTGCACCAACCAGCTGGGCATCGTGAAGTTCCTGCTGCAGAACTCCTGGCAGACGGCCGACATCAGCGCCAGGGACTCGGTGGGCAACACGGTGCTGCACGCCCTGGTGGAGGTGGCCGACAACACGGCCGACAACACGAAGTTTGTGACGAGCATGTACAATGAGATTCTGATCCTGGGGGCCAAACTGCACCCGACGCTGAAGCTGGAGGAGCTCACCAACAAGAAGGGAATGACGCCGCTGGCTCTGGCAGCTGGGACCGGGAAGATCGGGGTCTTGGCCTATATTCTCCAGCGGGAGATCCAGGAGCCCGAGTGCAGGCACCTGTCCAGGAAGTTCACCGAGTGGGCCTACGGGCCCGTGCACTCCTCGCTGTACGACCTGTCCTGCATCGACACCTGCGAGAAGAACTCGGTGCTGGAGGTGATCGCCTACAGCAGCAGCGAGACCCCTAATCGCCACGACATGCTCTTGGTGGAGCCGCTGAACCGACTCCTGCAGGACAAGTGGGACAGATTCGTCAAGCGCATCTTCTACTTCAACTTCCTGGTCTACTGCCTGTACATGATCATCTTCACCATGGCTGCCTACTACAGGCCCGTGGATGGCTTGCCTCCCTTTAAGATGGAAAAAACTGGAGACTATTTCCGAGTTACTGGAGAGATCCTGTCTGTGTTAGGAGGAGTCTACTTCTTTTTCCGAGGGATTCAGTATTTCCTGCAGAGGCGGCCGTCGATGAAGACCCTGTTTGTGGACAGCTACAGTGAGATGCTTTTCTTTCTGCAGTCACTGTTCATGCTGGCCACCGTGGTGCTGTACTTCAGCCACCTCAAGGAGTATGTGGCTTCCATGGTATTCTCCCTGGCCTTGGGCTGGACCAACATGCTCTACTACACCCGCGGTTTCCAGCAGATGGGCATCTATGCCGTCATGATAGAGAAGATGATCCTGAGAGACCTGTGCCGTTTCATGTTTGTCTACGTCGTCTTCTTGTTCGGGTTTTCCACAGCGGTGGTGACGCTGATTGAAGACGGGAAGAATGACTCCCTGCCGTCTGAGTCCACGTCGCACAGGTGGCGGGGGCCTGCCTGCAGGCCCCCCGATAGCTCCTACAACAGCCTGTACTCCACCTGCCTGGAGCTGTTCAAGTTCACCATCGGCATGGGCGACCTGGAGTTCACTGAGAACTATGACTTCAAGGCTGTCTTCATCATCCTGCTGCTGGCCTATGTAATTCTCACCTACATCCTCCTGCTCAACATGCTCATCGCCCTCATGGGTGAGACTGTCAACAAGATCGCACAGGAGAGCAAGAACATCTGGAAGCTGCAGAGAGCCATCACCATCCTGGACACGGAGAAGAGCTTCCTTAAGTGCATGAGGAAGGCCTTCCGCTCAGGCAAGCTGCTGCAGGTGGGGTACACACCTGATGGCAAGGACGACTACCGGTGGTGCTTCAGGGTGGACGAGGTGAACTGGACCACCTGGAACACCAACGTGGGCATCATCAACGAAGACCCGGGCAACTGTGAGGGCGTCAAGCGCACCCTGAGCTTCTCCCTGCGGTCAAGCAGAGTTTCAGGCAGACACTGGAAGAACTTTGCCCTGGTCCCCCTTTTAAGAGAGGCAAGTGCTCGAGATAGGCAGTCTGCTCAGCCCGAGGAAGTTTATCTGCGACAGTTTTCAGGGTCTCTGAAGCCAGAGGACGCTGAGGTCTTCAAGAGTCCTGCCGCTTCCGGGGAGAAGTGA

Protein sequence + ...

MKKWSSTDLGAAADPLQKDTCPDPLDGDPNSRPPPAKPQLSTAKSRTRLFGKGDSEEAFPVDCPHEEGELDSCPTITVSPVITIQRPGDGPTGARLLSQDSVAASTEKTLRLYDRRSIFEAVAQNNCQDLESLLLFLQKSKKHLTDNEFKDPETGKTCLLKAMLNLHDGQNTTIPLLLEIARQTDSLKELVNASYTDSYYKGQTALHIAIERRNMALVTLLVENGADVQAAAHGDFFKKTKGRPGFYFGELPLSLAACTNQLGIVKFLLQNSWQTADISARDSVGNTVLHALVEVADNTADNTKFVTSMYNEILILGAKLHPTLKLEELTNKKGMTPLALAAGTGKIGVLAYILQREIQEPECRHLSRKFTEWAYGPVHSSLYDLSCIDTCEKNSVLEVIAYSSSETPNRHDMLLVEPLNRLLQDKWDRFVKRIFYFNFLVYCLYMIIFTMAAYYRPVDGLPPFKMEKTGDYFRVTGEILSVLGGVYFFFRGIQYFLQRRPSMKTLFVDSYSEMLFFLQSLFMLATVVLYFSHLKEYVASMVFSLALGWTNMLYYTRGFQQMGIYAVMIEKMILRDLCRFMFVYIVFLFGFSTAVVTLIEDGKNDSLPSESTSHRWRGPACRPPDSSYNSLYSTCLELFKFTIGMGDLEFTENYDFKAVFIILLLAYVILTYILLLNMLIALMGETVNKIAQESKNIWKLQRAITILDTEKSFLKCMRKAFRSGKLLQVGYTPDGKDDYRWCFRVDEVNWTTWNTNVGIINEDPGNCEGVKRTLSFSLRSSRVSGRHWKNFALVPLLREASARDRQSAQPEEVYLRQFSGSLKPEDAEVFKSPAASGEK

GO Classification
component
intrinsic to membrane
integral to membrane
membrane
cell
function
transporter activity
ion transporter activity
ion channel activity
process
physiological process
cellular physiological process
transport
ion transport
See more information at   →   www.drugbank.ca
Id Name
DB00132 Alpha-Linolenic Acid
DB00159 Icosapent
DB00168 Aspartame
Id Name
DB00005 Etanercept
DB00035 Desmopressin
DB00041 Aldesleukin
DB00091 Cyclosporine
DB00132 Alpha-Linolenic Acid
DB00139 Succinic acid
DB00140 Riboflavin
DB00154 gamma-Homolinolenic acid
DB00158 Folic Acid
DB00159 Icosapent
DB00168 Aspartame
DB00175 Pravastatin
DB00181 Baclofen
DB00188 Bortezomib
DB00197 Troglitazone
DB00198 Oseltamivir
DB00214 Torasemide
DB00216 Eletriptan
DB00229 Cefotiam
DB00233 Aminosalicylic Acid
DB00244 Mesalazine
DB00250 Dapsone
DB00254 Doxycycline
DB00279 Liothyronine
DB00286 Conjugated Estrogens
DB00300 Tenofovir
DB00311 Ethoxzolamide
DB00313 Valproic Acid
DB00316 Acetaminophen
DB00319 Piperacillin
DB00327 Hydromorphone
DB00328 Indomethacin
DB00345 Aminohippurate
DB00350 Minoxidil
DB00360 Tetrahydrobiopterin
DB00365 Grepafloxacin
DB00369 Cidofovir
DB00374 Treprostinil
DB00390 Digoxin
DB00402 Eszopiclone
DB00412 Rosiglitazone
DB00425 Zolpidem
DB00432 Trifluridine
DB00437 Allopurinol
DB00438 Ceftazidime
DB00446 Chloramphenicol
DB00456 Cefalotin
DB00461 Nabumetone
DB00465 Ketorolac
DB00469 Tenoxicam
DB00470 Dronabinol
DB00471 Montelukast
DB00480 Lenalidomide
DB00482 Celecoxib
DB00493 Cefotaxime
DB00495 Zidovudine
DB00500 Tolmetin
DB00501 Cimetidine
DB00512 Vancomycin
DB00515 Cisplatin
DB00520 Caspofungin
DB00529 Foscarnet
DB00533 Rofecoxib
DB00536 Guanidine
DB00540 Nortriptyline
DB00549 Zafirlukast
DB00554 Piroxicam
DB00563 Methotrexate
DB00567 Cephalexin
DB00573 Fenoprofen
DB00577 Valaciclovir
DB00578 Carbenicillin
DB00580 Valdecoxib
DB00582 Voriconazole
DB00583 L-Carnitine
DB00584 Enalapril
DB00586 Diclofenac
DB00595 Oxytetracycline
DB00605 Sulindac
DB00606 Cyclothiazide
DB00607 Nafcillin
DB00619 Imatinib
DB00620 Triamcinolone
DB00624 Testosterone
DB00649 Stavudine
DB00672 Chlorpropamide
DB00678 Losartan
DB00693 Fluorescein
DB00695 Furosemide
DB00703 Methazolamide
DB00709 Lamivudine
DB00711 Diethylcarbamazine
DB00712 Flurbiprofen
DB00718 Adefovir Dipivoxil
DB00720 Clodronate
DB00731 Nateglinide
DB00744 Zileuton
DB00749 Etodolac
DB00759 Tetracycline
DB00773 Etoposide
DB00779 Nalidixic Acid
DB00783 Estradiol
DB00784 Mefenamic acid
DB00787 Acyclovir
DB00788 Naproxen
DB00795 Sulfasalazine
DB00796 Candesartan
DB00798 Gentamicin
DB00812 Phenylbutazone
DB00814 Meloxicam
DB00819 Acetazolamide
DB00821 Carprofen
DB00827 Cinoxacin
DB00829 Diazepam
DB00856 Chlorphenesin
DB00857 Terbinafine
DB00861 Diflunisal
DB00863 Ranitidine
DB00870 Suprofen
DB00880 Chlorothiazide
DB00884 Risedronate
DB00887 Bumetanide
DB00900 Didanosine
DB00903 Ethacrynic acid
DB00908 Quinidine
DB00912 Repaglinide
DB00917 Dinoprostone
DB00927 Famotidine
DB00936 Salicyclic acid
DB00939 Meclofenamic acid
DB00943 Zalcitabine
DB00945 Acetylsalicylic acid
DB00963 Bromfenac
DB00966 Telmisartan
DB00991 Oxaprozin
DB00999 Hydrochlorothiazide
DB01004 Ganciclovir
DB01009 Ketoprofen
DB01014 Balsalazide
DB01015 Sulfamethoxazole
DB01016 Glyburide
DB01017 Minocycline
DB01029 Irbesartan
DB01032 Probenecid
DB01033 Mercaptopurine
DB01041 Thalidomide
DB01050 Ibuprofen
DB01051 Novobiocin
DB01053 Penicillin G
DB01059 Norfloxacin
DB01060 Amoxicillin
DB01065 Melatonin
DB01067 Glipizide
DB01075 Diphenhydramine
DB01082 Streptomycin
DB01092 Ouabain
DB01124 Tolbutamide
DB01132 Pioglitazone
DB01136 Carvedilol
DB01137 Levofloxacin
DB01140 Cefadroxil
DB01147 Cloxacillin
DB01160 Dinoprost Tromethamine
DB01165 Ofloxacin
DB01181 Ifosfamide
DB01197 Captopril
DB01198 Zopiclone
DB01212 Ceftriaxone
DB01221 Ketamine
DB01237 Bromodiphenhydramine
DB01252 Mitiglinide
DB01283 Lumiracoxib
DB01326 Cefamandole
DB01327 Cefazolin
DB01329 Cefoperazone
DB01333 Cefradine
DB01355 Hexobarbital
DB01393 Bezafibrate
DB01395 Drospirenone
DB01397 Magnesium salicylate
DB01398 Salicylate-sodium
DB01399 Salsalate
DB01401 Trisalicylate-choline
DB01404 Ginseng
DB01414 Cefacetrile
DB01419 Antrafenine
DB01424 Aminophenazone
DB01435 Antipyrine
DB01583 Liotrix
DB01597 Cilastatin
DB01600 Tiaprofenic acid
DB01628 Etoricoxib
DB01650 trans-2-hydroxycinnamic acid
DB01837 O-Acetylserine
DB01892 Hyperforin
DB02047 2-(1,1'-Biphenyl-4-Yl)Propanoic Acid
DB02110 Protoporphyrin Ix Containing Co
DB02198 2-Bromoacetyl Group
DB02266 Flufenamic Acid
DB02315 Cyclic Guanosine Monophosphate
DB02379 Beta-D-Glucose
DB02527 Cyclic Adenosine Monophosphate
DB02659 Cholic Acid
DB02687 Beta-D-Mannose
DB02709 Resveratrol
DB02773 (3-Chloro-4-Propoxy-Phenyl)-Acetic Acid
DB02944 Alpha-D-Mannose
DB03014 Heme
DB03338 Heptyl-Beta-D-Glucopyranoside
DB03477 1-Phenylsulfonamide-3-Trifluoromethyl-5-Parabromophenylpyrazole
DB03553 Glutaric Acid
DB03585 Oxyphenbutazone
DB03667 Acetic Acid Salicyloyl-Amino-Ester
DB03752 P-(2'-Iodo-5'-Thenoyl)Hydrotropic Acid
DB03753 Flurbiprofen Methyl Ester
DB03756 Docosa-4,7,10,13,16,19-Hexaenoic Acid
DB03783 Phenacetin
DB03793 Benzoic Acid
DB03866 Prostaglandin G2
DB03902 Oxalic Acid
DB04133 Degraded Cephaloridine
DB04224 Oleic Acid
DB04270 (S)-3-(4-(2-Carbazol-9-Yl-Ethoxy)-Phenyl)-2-Ethoxy-Propionic Acid
DB04348 Taurocholic Acid
DB04519 Caprylic acid
DB04552 Niflumic Acid
DB04557 Arachidonic Acid
DB04689 2-{5-[3-(6-BENZOYL-1-PROPYLNAPHTHALEN-2-YLOXY)PROPOXY]INDOL-1-YL}ETHANOIC ACID
DB04743 Nimesulide
DB04801 (11E)-OCTADEC-11-ENOIC ACID
DB04817 Dipyrone
DB05109 Trabectedin
DB06151 Acetylcysteine
DB06335 Saxagliptin
DB06710 Methyltestosterone
DB06725 Lornoxicam
DB06802 Nepafenac
DB06804 Nonoxynol-9
DB06908 (2S)-3-(1-{[2-(2-CHLOROPHENYL)-5-METHYL-1,3-OXAZOL-4-YL]METHYL}-1H-INDOL-5-YL)-2-ETHOXYPROPANOIC ACID
DB06926 (9Z,11E,13S)-13-hydroxyoctadeca-9,11-dienoic acid
DB07053 2-{5-[3-(7-PROPYL-3-TRIFLUOROMETHYLBENZO[D]ISOXAZOL-6-YLOXY)PROPOXY]INDOL-1-YL}ETHANOIC ACID
DB07070 (2S)-2-{3-[({[2-fluoro-4-(trifluoromethyl)phenyl]carbonyl}amino)methyl]-4-methoxybenzyl}butanoic acid
DB07111 (4S,5E,7Z,10Z,13Z,16Z,19Z)-4-hydroxydocosa-5,7,10,13,16,19-hexaenoic acid
DB07172 (5R,6E,8Z,11Z,14Z,17Z)-5-hydroxyicosa-6,8,11,14,17-pentaenoic acid
DB07208 (8E,10S,12Z)-10-hydroxy-6-oxooctadeca-8,12-dienoic acid
DB07209 (8R,9Z,12Z)-8-hydroxy-6-oxooctadeca-9,12-dienoic acid
DB07302 (9S,10E,12Z)-9-hydroxyoctadeca-10,12-dienoic acid
DB07509 difluoro(5-{2-[(5-octyl-1H-pyrrol-2-yl-kappaN)methylidene]-2H-pyrrol-5-yl-kappaN}pentanoato)boron
DB07675 (2S)-2-ETHOXY-3-{4-[2-(10H-PHENOXAZIN-10-YL)ETHOXY]PHENYL}PROPANOIC ACID
DB07691 2-({[3-(3,4-dihydroisoquinolin-2(1H)-ylsulfonyl)phenyl]carbonyl}amino)benzoic acid
DB07723 3-(5-methoxy-1H-indol-3-yl)propanoic acid
DB07724 3-{5-methoxy-1-[(4-methoxyphenyl)sulfonyl]-1H-indol-3-yl}propanoic acid
DB07842 (2S)-2-(4-ethylphenoxy)-3-phenylpropanoic acid
DB07863 2-chloro-5-nitro-N-phenylbenzamide
DB07981 2-[1-(4-CHLOROBENZOYL)-5-METHOXY-2-METHYL-1H-INDOL-3-YL]-N-[(1R)-1-(HYDROXYMETHYL)PROPYL]ACETAMIDE
DB07983 1-(4-IODOBENZOYL)-5-METHOXY-2-METHYL INDOLE-3-ACETIC ACID
DB07984 2-[1-(4-CHLOROBENZOYL)-5-METHOXY-2-METHYL-1H-INDOL-3-YL]-N-[(1S)-1-(HYDROXYMETHYL)PROPYL]ACETAMIDE
DB08078 {4-[3-(4-acetyl-3-hydroxy-2-propylphenoxy)propoxy]phenoxy}acetic acid
DB08121 (2S)-2-(biphenyl-4-yloxy)-3-phenylpropanoic acid
DB08302 3-[5-(2-nitropent-1-en-1-yl)furan-2-yl]benzoic acid
DB08402 2-[(2,4-DICHLOROBENZOYL)AMINO]-5-(PYRIMIDIN-2-YLOXY)BENZOIC ACID
DB08435 (5E,14E)-11-oxoprosta-5,9,12,14-tetraen-1-oic acid
DB08560 3-FLUORO-N-[1-(4-FLUOROPHENYL)-3-(2-THIENYL)-1H-PYRAZOL-5-YL]BENZENESULFONAMIDE
DB08760 (2S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid
DB08814 Triflusal
DB08819 Tafluprost
DB08837 Tetraethylammonium
DB08846 Ellagic Acid
DB08910 Pomalidomide
DB08912 Dabrafenib
DB08915 ALEGLITAZAR